TargetRx Atlas

MRNA basic information

  • mRNA ID:ENST00000212015
  • Gene Name:SIRT1
  • mRNA database:Ensembl
  • mRNA expression :down-regulated
  • mRNA Method:PCR
  • mRNA Pathway:NA
  • Evidence:validated
  • (mRNA-drug)

Drug basic information

  • Drug ID:NA
  • Drug Name:Benzothiazepinone
  • Drug Method:down-regulated the gene expression

Disease basic infommation

  • Disease:acute lung injury
  • Tissue:patients tissues

Other information

  • Title:Discovery and anti-inflammatory evaluation of benzothiazepinones (BTZs) as novel non-ATP competitive inhibitors of glycogen synthase kinase-3β (GSK-3β)
  • Journal:Bioorganic & Medicinal Chemistry
  • Published:2018
  • PubMed ID:30293796
  • Abstract: